Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
YEATS domain-containing protein 2 (Homo sapiens) | BDBM50566877 (CHEMBL4863719) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.85E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00367 BindingDB Entry DOI: 10.7270/Q2833WSB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
YEATS domain-containing protein 2 (Homo sapiens) | BDBM50566890 (CHEMBL4865432) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00367 BindingDB Entry DOI: 10.7270/Q2833WSB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
YEATS domain-containing protein 2 (Homo sapiens) | BDBM50566867 (CHEMBL4855926) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00367 BindingDB Entry DOI: 10.7270/Q2833WSB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
YEATS domain-containing protein 2 (Homo sapiens) | BDBM50566873 (CHEMBL4859531) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00367 BindingDB Entry DOI: 10.7270/Q2833WSB | |||||||||||
More data for this Ligand-Target Pair |